SCHEMBL28451633

SCHEMBL28451633

OCC(CO)Nc1nc(Nc2cccc(C(F)(F)F)c2)nc(Oc2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 13/20 0.79
LMNA P02545 2/20 0.53
MAPT P10636 2/20 0.53
MAPK1 P28482 1/20 0.53
APP P05067 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28447648 0.89 IDH2 (1.00) IDH2LMNAMAPTMAPK1APP
SCHEMBL28450978 0.86 IDH2 (0.73) IDH2LMNAMAPTMAPK1APP
SCHEMBL28451527 0.85 IDH2 (0.71) IDH2LMNAMAPTMAPK1APP
SCHEMBL28451428 0.85 IDH2 (0.80) IDH2LMNAMAPTMAPK1APP
SCHEMBL28451427 0.85 IDH2 (0.80) IDH2LMNAMAPTMAPK1APP
SCHEMBL28457048 0.85 IDH2 (0.80) IDH2LMNAMAPTMAPK1APP
SCHEMBL28455014 0.83 IDH2 (0.88) IDH2LMNAMAPTMAPK1APP
SCHEMBL28450991 0.81 IDH2 (0.82) IDH2LMNAMAPTMAPK1APP
SCHEMBL28449181 0.80 IDH2 (0.79) IDH2LMNAMAPTMAPK1APP
SCHEMBL28450615 0.80 IDH2 (1.00) IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-B Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2023-10-24 CN disclosed
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed