SCHEMBL28455014

SCHEMBL28455014

OCC(CO)Nc1nc(Cl)nc(Nc2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.88

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 11/20 0.88
APP P05067 4/20 0.65
LMNA P02545 2/20 0.49
MAPT P10636 2/20 0.49
MAPK1 P28482 1/20 0.49
POLB P06746 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28447648 0.94 IDH2 (1.00) IDH2APPLMNAMAPTMAPK1
SCHEMBL28450991 0.85 IDH2 (0.82) IDH2APPLMNAMAPTMAPK1
SCHEMBL28450615 0.84 IDH2 (1.00) IDH2
SCHEMBL28451633 0.83 IDH2 (0.79) IDH2APPLMNAMAPTMAPK1
SCHEMBL30568814 0.83 APP (0.79) IDH2APPLMNAMAPTMAPK1
SCHEMBL1391344 0.83 APP (0.79) IDH2APPLMNAMAPTMAPK1
SCHEMBL28460991 0.83 IDH2 (0.89) IDH2APPLMNAMAPTMAPK1
SCHEMBL28451054 0.83 IDH2 (0.89) IDH2APPLMNAMAPTMAPK1
SCHEMBL28456839 0.83 IDH2 (0.89) IDH2APPLMNAMAPTMAPK1
SCHEMBL28459484 0.82 APP (0.65) IDH2APPLMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662242-B Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2023-10-24 CN disclosed
CN-111662242-A Heterocyclic IDH mutant inhibitor, preparation method and application thereof 中国药科大学 2020-09-15 CN disclosed