SCHEMBL28451900

SCHEMBL28451900

CCOC(=O)CCc1nc2cc(Cl)ccc2nc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.48
KDM4E B2RXH2 5/20 0.47
LMNA P02545 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 2/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
P2RY12 Q9H244 1/20 0.41
CYP4F2 P78329 2/20 0.40
CYP4A11 Q02928 2/20 0.40
PTPN1 P18031 1/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
RAB9A P51151 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28448193 1.00 EGFR (0.48) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28445478 0.88 EGFR (0.46) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28447306 0.88 EGFR (0.46) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28445383 0.87 KDM4E (0.61) KDM4ELMNAALDH1A1HSD17B10MAPT
SCHEMBL28454187 0.80 KDM4E (0.44) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28445422 0.80 KDM4E (0.44) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28452103 0.79 KDM4E (0.45) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28447304 0.79 KDM4E (0.45) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL28443132 0.79 MAPT (0.46) EGFRKDM4ELMNAALDH1A1HSD17B10
SCHEMBL17601553 0.76 GLP1R (0.51) KDM4EALDH1A1HSD17B10MAPTPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997230-B Quinoxaline derivative with matrix metalloproteinase inhibitory activity, preparation method and application thereof 山东大学 2020-08-04 CN disclosed