SCHEMBL28447306

SCHEMBL28447306

CCOC(=O)CCc1nc2cc(Br)ccc2nc1Cl

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 3/20 0.46
LMNA P02545 2/20 0.46
HSD17B10 Q99714 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 3/20 0.40
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
P2RY12 Q9H244 1/20 0.39
CYP4F2 P78329 2/20 0.39
CYP4A11 Q02928 2/20 0.39
ATM Q13315 2/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28445478 1.00 EGFR (0.46) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL28451900 0.88 EGFR (0.48) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL28448193 0.88 EGFR (0.48) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL9378 0.88 EGFR (0.60) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL28445383 0.84 KDM4E (0.61) ALDH1A1KDM4ELMNAHSD17B10SMN1; SMN2
SCHEMBL9365 0.82 HDAC6 (0.43) EGFRALDH1A1KDM4EMAPTGLA
SCHEMBL28443100 0.78 KDM4E (0.44) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL28445463 0.77 ALDH1A1 (0.43) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL28451603 0.77 ALDH1A1 (0.43) EGFRALDH1A1KDM4ELMNAHSD17B10
SCHEMBL28449192 0.76 KDM4E (0.71) EGFRALDH1A1KDM4ELMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997230-B Quinoxaline derivative with matrix metalloproteinase inhibitory activity, preparation method and application thereof 山东大学 2020-08-04 CN disclosed