SCHEMBL28453154

SCHEMBL28453154

COc1cc(C(=O)O)cc(N)c1NCC=CCNC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 1/20 0.38
NR1H4 Q96RI1 2/20 0.36
EPHX2 P34913 1/20 0.36
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA4 P22748 2/20 0.36
CA6 P23280 2/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
CA14 Q9ULX7 2/20 0.36
CA3 P07451 1/20 0.36
PKM P14618 1/20 0.36
CA5A P35218 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
PTGS2 P35354 1/20 0.35
CNR2 P34972 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28453150 1.00 STING1 (0.38) STING1NR1H4EPHX2CA12CA1
SCHEMBL29080502 0.91 STING1 (0.38) STING1CNR2ALDH1A1LMNAHTT
SCHEMBL20889072 0.91 STING1 (0.45) STING1ALDH1A1LMNAHTTL3MBTL1
SCHEMBL22313218 0.91 STING1 (0.38) STING1CNR2ALDH1A1LMNAHTT
SCHEMBL29012734 0.91 STING1 (0.45) STING1ALDH1A1LMNAHTTL3MBTL1
SCHEMBL29406354 0.91 STING1 (0.45) STING1ALDH1A1LMNAHTTL3MBTL1
SCHEMBL28880366 0.83 MAPT (0.42) ALDH1A1LMNATPMTMAPTMEN1
SCHEMBL25098877 0.81 STING1 (0.46) STING1CA12CA1CA2CA9
SCHEMBL29868394 0.81 STING1 (0.46) STING1CA12CA1CA2CA9
SCHEMBL22519927 0.81 DRD2 (0.41) EPHX2CA1CA2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113563313-B Immunomodulator 成都先导药物开发股份有限公司 2022-11-04 CN disclosed
CN-113563313-A Immunomodulator 成都先导药物开发股份有限公司 2021-10-29 CN disclosed
CN-111499617-B Immunomodulator 成都先导药物开发股份有限公司 2021-08-06 CN disclosed
CN-111499617-A Immunomodulator 成都先导药物开发股份有限公司 2020-08-07 CN disclosed