SCHEMBL28456342

SCHEMBL28456342

CC(C)(C)OC(=O)N1CC(n2cc3cc(Br)ccc3n2)C1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.44
FPR2 P25090 4/20 0.42
BACE1 P56817 2/20 0.39
RORC P51449 2/20 0.39
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SSTR4 P31391 1/20 0.38
FPR3 P25089 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36
TLR8 Q9NR97 1/20 0.36
JAK1 P23458 1/20 0.36
KRAS P01116 2/20 0.35
PDE4B Q07343 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29042019 0.91 USP30 (0.47) USP30FPR2BACE1GPR119ABL1
SCHEMBL29042052 0.91 USP30 (0.47) USP30FPR2BACE1GPR119ABL1
SCHEMBL28457723 0.91 USP30 (0.44) USP30FPR2BACE1RORCKCNK3
SCHEMBL28463632 0.90 FPR2 (0.48) USP30FPR2BACE1FPR3JAK1
SCHEMBL20135633 0.89 FPR2 (0.45) USP30FPR2BACE1GPR119
SCHEMBL25335635 0.83 USP30 (0.43) USP30FPR2BACE1RORCKCNK3
SCHEMBL25958972 0.83 USP30 (0.43) USP30FPR2BACE1RORCKCNK3
SCHEMBL25335630 0.83 USP30 (0.43) USP30FPR2BACE1RORCKCNK3
SCHEMBL26654669 0.81 EHMT2 (0.43) PDE4B
SCHEMBL28456256 0.81 FPR2 (0.48) USP30FPR2BACE1FPR3JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117986262-A Condensed bicyclic compounds, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2024-05-07 CN disclosed
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed