SCHEMBL28457906

SCHEMBL28457906

C1CCOCC1.Nc1ccc2ccsc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
GAA P10253 3/20 0.39
RAB9A P51151 3/20 0.39
NPC1 O15118 2/20 0.39
KDM4E B2RXH2 2/20 0.39
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CA2 P00918 1/20 0.33
DYRK1A Q13627 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 1/20 0.33
CYP2A6 P11509 1/20 0.32
SIGMAR1 Q99720 1/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA7 P36544 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL397816 0.84 ALDH1A1 (0.42) MAPTSMN1; SMN2GAARAB9ANPC1
Hydrochloric Acid SCHEMBL15880793 0.82 ALDH1A1 (0.41) MAPTSMN1; SMN2GAARAB9ANPC1
Benzothiophene SCHEMBL28919762 0.75 CTNNB1 (0.35) SMN1; SMN2RAB9ANPC1KDM4ESLC6A2
SCHEMBL760406 0.68 CYP2A6 (0.55) MAPTGAARAB9ANPC1KDM4E
SCHEMBL826863 0.67 CYP2A6 (0.42) MAPTRAB9AKDM4ESLC6A2SLC6A4
SCHEMBL19756637 0.67 SLC6A4 (0.43) SLC6A2SLC6A4SLC6A3HTR3EHTR3B
SCHEMBL19756623 0.67 SLC6A2 (0.57) MAPTSMN1; SMN2RAB9ANPC1KDM4E
Hydrochloric Acid SCHEMBL10370258 0.66 CYP2A6 (0.53) MAPTGAARAB9ANPC1KDM4E
SCHEMBL17449212 0.65 MAPT (0.44) MAPTSMN1; SMN2GAARAB9ANPC1
SCHEMBL17449204 0.65 MAPT (0.44) MAPTSMN1; SMN2GAARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111658644-B Small-molecule STAT3 inhibitor WZ-2-033 and application thereof in preparation of medicines for treating breast cancer and gastric cancer 中山大学 2021-05-14 CN disclosed
CN-111658644-A Small-molecule STAT3 inhibitor WZ-2-033 and application thereof in preparation of medicines for treating breast cancer and gastric cancer 中山大学 2020-09-15 CN disclosed