SCHEMBL28458754

SCHEMBL28458754

CN(c1ncnc2[nH]ccc12)C1CCN(CC(=O)Nc2ccccc2Cl)CC1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 18/20 0.56
JAK2 O60674 13/20 0.56
JAK3 P52333 8/20 0.52
TYK2 P29597 3/20 0.51
KCNH2 Q12809 1/20 0.51
BTK Q06187 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28463172 0.88 JAK1 (0.54) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28459247 0.86 JAK1 (0.68) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28458823 0.83 GRIN2B (0.55) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28468658 0.81 PAK1 (0.57) KCNH2BTK
SCHEMBL3537591 0.78 JAK1 (0.73) JAK1JAK2JAK3TYK2
SCHEMBL28460152 0.77 JAK1 (0.61) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28468948 0.77 JAK1 (0.66) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28899230 0.76 JAK1 (0.65) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28462184 0.75 JAK1 (0.64) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL21400284 0.75 JAK1 (0.76) JAK1JAK2JAK3TYK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111620873-A Pyrrolo [2,3-d ] pyrimidine derivatives containing piperidine and preparation and application thereof 沈阳药科大学 2020-09-04 CN claimed
CN-111620873-B Pyrrolo [2,3-d ] pyrimidine derivatives containing piperidine and preparation and application thereof 沈阳药科大学 2021-12-28 CN disclosed
CN-111620873-A Pyrrolo [2,3-d ] pyrimidine derivatives containing piperidine and preparation and application thereof 沈阳药科大学 2020-09-04 CN disclosed