SCHEMBL28459247

SCHEMBL28459247

CN(c1ncnc2[nH]ccc12)C1CCN(C(=O)Nc2ccccc2Cl)CC1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 17/20 0.68
JAK2 O60674 13/20 0.68
JAK3 P52333 6/20 0.56
TYK2 P29597 1/20 0.56
KCNH2 Q12809 1/20 0.56
BTK Q06187 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28458754 0.86 JAK1 (0.56) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL21400612 0.84 JAK2 (0.71) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28466426 0.83 JAK1 (0.62) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL20183394 0.81 JAK1 (1.00) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL20183389 0.81 JAK1 (1.00) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL21400284 0.81 JAK1 (0.76) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL21400276 0.81 JAK1 (0.76) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL28465851 0.80 PAK1 (0.76) JAK1JAK2JAK3BTK
SCHEMBL21400293 0.79 JAK1 (0.60) JAK1JAK2JAK3TYK2KCNH2
SCHEMBL21400286 0.79 JAK1 (0.71) JAK1JAK2JAK3TYK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111620873-A Pyrrolo [2,3-d ] pyrimidine derivatives containing piperidine and preparation and application thereof 沈阳药科大学 2020-09-04 CN claimed
CN-111620873-B Pyrrolo [2,3-d ] pyrimidine derivatives containing piperidine and preparation and application thereof 沈阳药科大学 2021-12-28 CN disclosed
CN-111620873-A Pyrrolo [2,3-d ] pyrimidine derivatives containing piperidine and preparation and application thereof 沈阳药科大学 2020-09-04 CN disclosed