SCHEMBL28458968

SCHEMBL28458968

N#Cc1ccc([C@H]2CO2)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.45
CYP11B1 P15538 3/20 0.45
CYP19A1 P11511 2/20 0.45
CYP17A1 P05093 1/20 0.45
HRH1 P35367 1/20 0.45
KCNH2 Q12809 1/20 0.45
CHRNA1 P02708 1/20 0.40
CHRNG P07510 1/20 0.40
CHRNB1 P11230 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
CHRND Q07001 1/20 0.40
CYP2D6 P10635 1/20 0.39
GSK3B P49841 1/20 0.39
DPP4 P27487 4/20 0.38
DRD2 P14416 3/20 0.35
DRD3 P35462 3/20 0.35
ELANE P08246 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31160051 1.00 CYP11B2 (0.45) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL10687001 0.81 GRM2 (0.42) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL10687012 0.81 GRM2 (0.42) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL10687018 0.81 GRM2 (0.42) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL122002 0.78 CYP11B2 (0.43) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL31140530 0.78 MAPT (0.41) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL10501106 0.76 CYP11B2 (0.39) CYP11B2CYP11B1CYP19A1CYP17A1HRH1
SCHEMBL1121711 0.75 HTR2A (0.49) CHRNB2CHRNB4CHRNA3CHRNA4DPP4
SCHEMBL12303672 0.75 HTR2A (0.49) CHRNB2CHRNB4CHRNA3CHRNA4DPP4
SCHEMBL29595508 0.75 HTR2A (0.49) CHRNB2CHRNB4CHRNA3CHRNA4DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111517985-B Preparation method of 4- [ (1R) -1-amino-2-hydroxyethyl ] -3-fluoro-benzonitrile 济南百润医药科技有限公司 2023-05-12 CN claimed
CN-111517985-A Preparation method of 4- [ (1R) -1-amino-2-hydroxyethyl ] -3-fluoro-benzonitrile 苏州明锐医药科技有限公司 2020-08-11 CN claimed
CN-111517985-B Preparation method of 4- [ (1R) -1-amino-2-hydroxyethyl ] -3-fluoro-benzonitrile 济南百润医药科技有限公司 2023-05-12 CN disclosed