SCHEMBL28459503

SCHEMBL28459503

Cc1cccc(-c2cncn2C(c2ccccc2)(c2ccccc2)c2ccccc2)c1C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.36
P2RX7 Q99572 4/20 0.35
IDO1 P14902 6/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
TDO2 P48775 2/20 0.32
LMNA P02545 1/20 0.32
LCK P06239 1/20 0.32
SRC P12931 1/20 0.32
LDLR P01130 1/20 0.31
PCSK9 Q8NBP7 1/20 0.31
HPGDS O60760 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20225762 0.75 FYN (0.32) IDO1CYP11B1CYP11B2
SCHEMBL19732321 0.73 IDO1 (0.57) NUDT1P2RX7IDO1CYP11B1CYP11B2
SCHEMBL1484285 0.73 GAA (0.36) IDO1CYP11B1CYP11B2HSP90AA1HSP90AB1
SCHEMBL4806085 0.73 CYP11B1 (0.43) P2RX7CYP11B1CYP11B2HSP90AA1LMNA
SCHEMBL1482948 0.72 KMT2A (0.37) LMNAALDH1A1
SCHEMBL1638486 0.72 CYP19A1 (0.37) CYP11B1CYP11B2LMNAALDH1A1
SCHEMBL2205776 0.72 CYP19A1 (0.32) CYP11B1CYP11B2LMNA
SCHEMBL20225761 0.71 NPC1 (0.36) IDO1LMNALCKALDH1A1
SCHEMBL1639289 0.70 CYP46A1 (0.36) CYP11B1CYP11B2LMNALCKSRC
SCHEMBL1482976 0.69 GAA (0.35) IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107879979-B Preparation method of dexmedetomidine 广东莱佛士制药技术有限公司 2020-08-25 CN claimed
CN-107879979-B Preparation method of dexmedetomidine 广东莱佛士制药技术有限公司 2020-08-25 CN disclosed
CN-107879979-B Preparation method of dexmedetomidine 广东莱佛士制药技术有限公司 2020-08-25 CN disclosed