SCHEMBL4806085

SCHEMBL4806085

Cc1cncn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.43
CYP11B2 P19099 3/20 0.43
CYP19A1 P11511 3/20 0.35
KCNN4 O15554 3/20 0.35
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
NR1I2 O75469 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
TBXA2R P21731 2/20 0.35
CCKBR P32239 2/20 0.35
OPRK1 P41145 2/20 0.35
SLC6A3 Q01959 2/20 0.35
KCNH2 Q12809 2/20 0.35
NR1H4 Q96RI1 2/20 0.35
MAPK1 P28482 2/20 0.35
MEN1 O00255 1/20 0.35
SLC22A1 O15245 1/20 0.35
GMNN O75496 1/20 0.35
USP2 O75604 1/20 0.35
TRPM2 O94759 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11750663 0.78 CYP11B1 (0.35) CYP11B1CYP11B2CYP19A1CHRM2CYP3A4
SCHEMBL11891094 0.78 ALDH1A1 (0.41) CYP11B1CYP11B2KCNN4MAPK1ABCB11
SCHEMBL2204500 0.77 CYP11B1 (0.43) CYP11B1CYP11B2CYP19A1KCNN4MAOA
SCHEMBL16371592 0.77 CYP11B1 (0.47) CYP11B1CYP11B2CYP19A1KCNN4MAOA
SCHEMBL27638465 0.77 CYP11B1 (0.43) CYP11B1CYP11B2CYP19A1KCNN4MAOA
SCHEMBL11891091 0.75 CYP11B1 (0.39) CYP11B1CYP11B2CYP19A1KCNN4MAOA
SCHEMBL12267644 0.74 TDP1 (0.35) CYP11B1CYP11B2CYP19A1LMNACYP3A4
SCHEMBL11891093 0.74 CYP11B1 (0.38) CYP11B1CYP11B2CYP19A1KCNN4MAOA
SCHEMBL28459503 0.73 NUDT1 (0.36) CYP11B1CYP11B2LMNALDLRPCSK9
SCHEMBL25190881 0.73 CYP11B1 (0.40) CYP11B1CYP11B2CYP19A1KCNN4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344619-B1 PHENOXYMETHYL DERIVATIVES HOFFMANN LA ROCHE (CH) 2020-10-28 EP disclosed
WO-2017037146-A1 PHENOXYMETHYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2017-03-09 WO disclosed
WO-2008088937-A1 QUINOLYNYLMETHYLIMIDIZOLES AS THERAPEUTIC AGENTS ALLERGAN, INC. (US) 2008-07-24 WO disclosed