SCHEMBL28461533

SCHEMBL28461533

C=C/C=C/C(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N1CC(N(C)C)C1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.70
IGF1R P08069 4/20 0.65
KCNH2 Q12809 4/20 0.65
INSR P06213 2/20 0.65
CCNT1 O60563 2/20 0.55
CCNA2 P20248 2/20 0.55
CDK2 P24941 2/20 0.55
CDK7 P50613 2/20 0.55
CDK9 P50750 2/20 0.55
CCNH P51946 2/20 0.55
MNAT1 P51948 1/20 0.55
CCNK O75909 1/20 0.54
CDK13 Q14004 1/20 0.54
CDK12 Q9NYV4 1/20 0.54
ALK Q9UM73 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28942037 1.00 EGFR (0.70) EGFRIGF1RKCNH2INSRCCNT1
SCHEMBL28942042 0.95 EGFR (0.69) EGFRIGF1RKCNH2INSRCCNT1
SCHEMBL28469195 0.95 EGFR (0.69) EGFRIGF1RKCNH2INSRCCNT1
SCHEMBL14719276 0.94 EGFR (0.80) EGFRIGF1RKCNH2INSRCCNT1
SCHEMBL28942024 0.90 EGFR (0.87) EGFRIGF1RKCNH2CCNT1CCNA2
SCHEMBL28467425 0.90 EGFR (0.87) EGFRIGF1RKCNH2CCNT1CCNA2
SCHEMBL14718460 0.89 EGFR (0.79) EGFRIGF1RKCNH2INSRCCNT1
SCHEMBL28942052 0.88 EGFR (0.67) EGFRIGF1RKCNH2INSR
SCHEMBL28467428 0.88 EGFR (0.67) EGFRIGF1RKCNH2INSR
SCHEMBL28470066 0.88 EGFR (0.70) EGFRIGF1RKCNH2INSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191861-B N- [5- (pyrimidin-2-amino) -2, 4-disubstituted-phenyl ] -trans-2, 4-pentadiene-amide 天津大学 2020-10-02 CN disclosed