SCHEMBL28462255

SCHEMBL28462255

[2H]C([2H])([2H])C(F)(C[C@H]1COC(=O)N1)C([2H])([2H])[2H]

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 5/20 0.33
HTR1B P28222 5/20 0.33
HTR1A P08908 2/20 0.33
KMT2A Q03164 1/20 0.33
HTR2A P28223 1/20 0.33
ADRA1A P35348 1/20 0.33
KCNH2 Q12809 1/20 0.32
CACNA1C Q13936 1/20 0.32
SCN5A Q14524 1/20 0.32
HTR1F P30939 1/20 0.32
AR P10275 2/20 0.32
IRAK4 Q9NWZ3 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28462259 1.00 HTR1D (0.33) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL15905687 0.95 HTR1D (0.32) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL5170319 0.88 KCNH2 (0.33) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL2155869 0.88 KCNH2 (0.33) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL24324048 0.88 KCNH2 (0.33) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL28469014 0.80 HTR1D (0.33) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL28469012 0.80 HTR1D (0.33) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL15905689 0.79 HTR1D (0.32) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL8873531 0.77 PLG (0.34) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL8873526 0.77 PLG (0.34) HTR1DHTR1BHTR1AKMT2AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106866502-B Cathepsin K inhibitors and uses thereof 广东东阳光药业有限公司 2020-10-09 CN disclosed