SCHEMBL28463263

SCHEMBL28463263

CCOC(=O)c1cc2c(NCc3ccccc3)ccc([N+](=O)[O-])c2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 15/20 0.55
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
USP2 O75604 1/20 0.45
HTT P42858 1/20 0.45
RECQL P46063 1/20 0.45
MAPT P10636 2/20 0.45
CRHBP P24387 2/20 0.45
CRHR2 Q13324 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28455858 0.90 FBP1 (0.69) FBP1MEN1KMT2AMAPTCRHBP
SCHEMBL28469977 0.86 FBP1 (0.66) FBP1
SCHEMBL28461385 0.85 FBP1 (0.62) FBP1KMT2AMAPTCRHBPCRHR2
SCHEMBL28469953 0.84 FBP1 (0.62) FBP1KMT2AHTTMAPTNPC1
SCHEMBL28463835 0.83 FBP1 (0.64) FBP1MAPTCRHBPCRHR2NPC1
SCHEMBL28469967 0.82 FBP1 (0.53) FBP1MEN1KMT2AMAPTNPC1
SCHEMBL28467678 0.82 FBP1 (0.67) FBP1
SCHEMBL28457753 0.81 FBP1 (0.52) FBP1
SCHEMBL28461240 0.81 FBP1 (0.65) FBP1MAPTCRHBPCRHR2NPC1
SCHEMBL28467759 0.80 FBP1 (0.66) FBP1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098846-B N-acyl sulfonamide FBPase inhibitor, preparation method thereof, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-10-09 CN disclosed