SCHEMBL28464628

SCHEMBL28464628

CCc1nn2ccc(C)cc2c1C(=O)c1cc(Br)c(O)c(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 11/20 0.42
TTR P02766 5/20 0.40
EYA3 Q99504 4/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
HPGD P15428 2/20 0.40
ESR1 P03372 2/20 0.40
EYA2 O00167 1/20 0.40
MEN1 O00255 1/20 0.40
ABCC4 O15439 1/20 0.40
PLIN1 O60240 1/20 0.40
NR1I2 O75469 1/20 0.40
USP2 O75604 1/20 0.40
ABCB11 O95342 1/20 0.40
ALB P02768 1/20 0.40
NR3C1 P04150 1/20 0.40
CYP1A2 P05177 1/20 0.40
PGR P06401 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20181603 0.84 SLC22A12 (0.46) SLC22A12TTREYA3CYP2C9CYP2C19
SCHEMBL24592873 0.84 SLC22A12 (0.38) SLC22A12EYA3CYP2C9ALDH1A1LMNA
SCHEMBL28464553 0.81 SLC22A12 (0.41) SLC22A12TTREYA3CYP2C9CYP2C19
SCHEMBL28468102 0.78 SLC22A12 (0.41) SLC22A12TTREYA3CYP2C9CYP2C19
SCHEMBL28467063 0.77 TTR (0.43) SLC22A12TTREYA3CYP2C9CYP2C19
SCHEMBL19531525 0.76 KDM4E (0.44) ALDH1A1HPGDMEN1POLBADORA3
SCHEMBL28470517 0.76 SLC22A12 (0.49) SLC22A12TTREYA3CYP2C9CYP2C19
SCHEMBL28462692 0.75 TTR (0.44) SLC22A12TTREYA3CYP2C9CYP2C19
SCHEMBL21584617 0.70 PTGDR2 (0.37) SLC22A12CYP2C9CYP2C19ALDH1A1MEN1
SCHEMBL21584605 0.69 ELANE (0.41) ALDH1A1LMNAADORA3MAPTPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107759588-B Phenyl- (pyrazolo [1,5-a ] pyridine-3-yl) ketone derivative 江苏新元素医药科技有限公司 2020-10-23 CN claimed
CN-107759588-B Phenyl- (pyrazolo [1,5-a ] pyridine-3-yl) ketone derivative 江苏新元素医药科技有限公司 2020-10-23 CN disclosed