SCHEMBL28464641

SCHEMBL28464641

CSc1ncc(C(=O)Cl)c(Br)n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
AHR P35869 1/20 0.43
MAPT P10636 3/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
THRB P10828 2/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 2/20 0.37
HPGD P15428 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22056908 0.84 MEN1 (0.51) MEN1KMT2AAHRMAPTNPC1
SCHEMBL5656811 0.81 MEN1 (0.51) MEN1KMT2AAHRMAPTNPC1
SCHEMBL22056715 0.80 ALDH1A1 (0.46) MEN1KMT2AAHRMAPTNPC1
SCHEMBL8399451 0.78 POLB (0.51) MEN1KMT2AAHRMAPTTHRB
SCHEMBL4572858 0.77 MEN1 (0.44) MEN1KMT2AAHRMAPTNPC1
SCHEMBL29776216 0.76 KMT2A (0.54) MEN1KMT2AAHRMAPTNPC1
SCHEMBL10517153 0.76 KMT2A (0.54) MEN1KMT2AAHRMAPTNPC1
SCHEMBL3970809 0.73 AHR (0.41) MEN1KMT2AAHRMAPTNPC1
SCHEMBL28463061 0.71 MAPT (0.52) MEN1KMT2AMAPTTHRBALDH1A1
SCHEMBL6039621 0.70 KMT2A (0.75) MEN1KMT2AMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109553607-B Pyrimidine carboxamide derivatives, preparation method, composition, preparation and application thereof 镇江圣安医药有限公司 2020-09-01 CN claimed
CN-109553607-B Pyrimidine carboxamide derivatives, preparation method, composition, preparation and application thereof 镇江圣安医药有限公司 2020-09-01 CN disclosed