SCHEMBL28465845

SCHEMBL28465845

COc1cc2ncnc(Oc3cc(F)c(C(=O)C(=O)Nc4ccc(C#N)c(C(F)(F)F)c4)c(F)c3)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRAF P15056 11/20 0.57
RAF1 P04049 6/20 0.57
KDR P35968 9/20 0.53
MAPK14 Q16539 1/20 0.51
TNNI3K Q59H18 1/20 0.51
PDGFRA P16234 1/20 0.51
EGFR P00533 1/20 0.51
MET P08581 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28900928 0.88 BRAF (0.70) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL28473758 0.86 KDR (0.59) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL28979425 0.85 BRAF (0.56) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL30447912 0.85 BRAF (0.56) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL28464544 0.84 BRAF (0.51) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL30447715 0.84 KDR (0.71) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL30448158 0.83 MET (0.65) BRAFRAF1KDRPDGFRAMET
SCHEMBL30447998 0.83 BRAF (0.57) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL30448378 0.83 BRAF (0.72) BRAFRAF1KDRMAPK14TNNI3K
SCHEMBL30448305 0.83 BRAF (0.61) BRAFRAF1KDRMAPK14TNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825605-B Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2023-03-31 CN disclosed
CN-111825605-A Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2020-10-27 CN disclosed