SCHEMBL28469729

SCHEMBL28469729

Cc1c(Nc2ccc(N(C)C)cc2)nc2ccccc2c1C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 18/20 0.64
KDM4E B2RXH2 1/20 0.57
MEN1 O00255 1/20 0.57
USP2 O75604 1/20 0.57
LMNA P02545 1/20 0.57
TP53 P04637 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
MAPT P10636 1/20 0.57
CYP2C9 P11712 1/20 0.57
HPGD P15428 1/20 0.57
TSHR P16473 1/20 0.57
MAPK1 P28482 1/20 0.57
CYP2C19 P33261 1/20 0.57
RECQL P46063 1/20 0.57
KMT2A Q03164 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
NPC1 O15118 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28469640 0.85 KDM1A (0.67) KDM1AMEN1USP2LMNATP53
SCHEMBL28481400 0.84 NPY5R (0.63) KDM1AKDM4EMEN1LMNATP53
SCHEMBL28478208 0.83 ABCG2 (0.56) KDM1AKDM4EMEN1LMNATP53
SCHEMBL2258103 0.82 KDM1A (0.71) KDM1AKDM4EMEN1USP2LMNA
SCHEMBL3347553 0.78 KDM1A (1.00) KDM1A
SCHEMBL8908702 0.78 NPY5R (0.74) KDM1ANPC1PKMRAB9AKLF5
SCHEMBL28468206 0.78 ABCG2 (0.61) KDM1AKDM4EMEN1LMNATP53
SCHEMBL29569079 0.78 MAPT (0.57) KDM1AMEN1TP53MAPTKMT2A
SCHEMBL12993921 0.78 MAPT (0.57) KDM1AMEN1TP53MAPTKMT2A
Hydrochloric Acid SCHEMBL8900394 0.77 NPY5R (0.72) KDM1ANPC1PKMRAB9AKLF5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116143693-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-05-23 CN claimed
CN-111825610-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2020-10-27 CN claimed
CN-116143693-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-05-23 CN disclosed
CN-111825610-B 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-03-31 CN disclosed
CN-111825610-A 2-methylquinoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2020-10-27 CN disclosed