SCHEMBL28470533

SCHEMBL28470533

COc1cc2ncnc(Oc3ccc(C(=O)C(=O)O)c(O)c3)c2cc1OC

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.63
RET P07949 1/20 0.63
KIF5B P33176 1/20 0.63
CSF1R P07333 1/20 0.58
AURKA O14965 1/20 0.58
MET P08581 1/20 0.58
TEK Q02763 1/20 0.58
AURKB Q96GD4 1/20 0.58
PDGFRA P16234 1/20 0.57
BRAF P15056 2/20 0.56
EGFR P00533 3/20 0.55
RAF1 P04049 1/20 0.54
LCK P06239 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30447669 0.88 KDR (0.65) KDRRETKIF5BCSF1RAURKA
SCHEMBL28474019 0.88 KDR (0.65) KDRRETKIF5BCSF1RAURKA
SCHEMBL30447427 0.86 KDR (0.62) KDRRETKIF5BCSF1RAURKA
SCHEMBL28475707 0.86 KDR (0.62) KDRRETKIF5BCSF1RAURKA
SCHEMBL28468402 0.84 KDR (0.66) KDRRETKIF5BCSF1RAURKA
SCHEMBL30447769 0.84 KDR (0.66) KDRRETKIF5BCSF1RAURKA
SCHEMBL28464516 0.83 PDGFRA (0.62) KDRAURKAMETTEKAURKB
SCHEMBL30448190 0.83 PDGFRA (0.62) KDRAURKAMETTEKAURKB
SCHEMBL5959059 0.81 KDR (0.71) KDRRETKIF5BCSF1RAURKA
SCHEMBL4365791 0.81 KDR (0.74) KDRRETKIF5BCSF1RPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111825605-A Aryl ketone amide compound and preparation method and application thereof 中国科学院上海药物研究所 2020-10-27 CN disclosed