SCHEMBL28474337

SCHEMBL28474337

c1ccc(-c2nc(-c3ccnc4ccccc34)nc3ccccc23)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.58
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
ATM Q13315 1/20 0.54
ADORA2A P29274 2/20 0.50
TGFBR1 P36897 2/20 0.49
MAPK14 Q16539 2/20 0.49
NUDT1 P36639 3/20 0.49
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 3/20 0.45
HPGD P15428 2/20 0.45
NPC1 O15118 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPT P10636 3/20 0.45
GAA P10253 1/20 0.45
HTR2B P41595 1/20 0.44
MTNR1A P48039 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16436780 0.88 MEN1 (0.59) CYP1A2MEN1KMT2AATMADORA2A
SCHEMBL17412545 0.86 MEN1 (0.64) MEN1KMT2AATMADORA2ANUDT1
SCHEMBL24589733 0.84 METAP1 (0.52) CYP1A2MEN1KMT2ATGFBR1MAPK14
SCHEMBL13911018 0.83 MEN1 (0.64) MEN1KMT2AATMADORA2ANUDT1
SCHEMBL24589842 0.81 TSHR (0.49) CYP1A2MEN1KMT2ATGFBR1MAPK14
SCHEMBL9920500 0.80 MEN1 (0.70) MEN1KMT2AATMADORA2ANUDT1
SCHEMBL15940567 0.80 L3MBTL1 (0.53) CYP1A2MEN1KMT2AADORA2ATGFBR1
SCHEMBL21131884 0.79 CYP1A2 (0.53) CYP1A2MEN1KMT2AATMTGFBR1
SCHEMBL4499365 0.79 CYP1A2 (0.54) CYP1A2ADORA2ATGFBR1MAPK14ALDH1A1
SCHEMBL2913642 0.79 METAP1 (0.64) MEN1KMT2AATMALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111700894-B Application of 2-azaarene substituted quinazoline compound in preparation of antitumor drugs 南方医科大学 2023-07-28 CN disclosed
CN-111700894-A Application of 2-azaarene substituted quinazoline compound in preparation of antitumor drugs 南方医科大学 2020-09-25 CN disclosed