SCHEMBL28475201

SCHEMBL28475201

Nc1ccccc1NC(=O)C=Cc1ccc(NC(=O)c2ccc(N(CCCl)CCCl)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 0.55
NAMPT P43490 1/20 0.55
EGFR P00533 2/20 0.51
ERBB2 P04626 2/20 0.51
HDAC3 O15379 3/20 0.50
HDAC2 Q92769 3/20 0.50
HDAC8 Q9BY41 2/20 0.50
NCOR1 O75376 1/20 0.50
HDAC4 P56524 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
NCOR2 Q9Y618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28468321 0.87 EGFR (0.65) HDAC1EGFRERBB2HDAC3HDAC2
SCHEMBL28468900 0.84 EGFR (0.59) HDAC1EGFRERBB2HDAC3HDAC2
SCHEMBL28469673 0.84 EGFR (0.69) HDAC1EGFRERBB2HDAC3HDAC2
SCHEMBL1064701 0.81 HDAC1 (0.65) HDAC1NAMPTHDAC3HDAC2HDAC8
SCHEMBL1064700 0.81 HDAC1 (0.65) HDAC1NAMPTHDAC3HDAC2HDAC8
SCHEMBL28477425 0.81 EGFR (0.60) HDAC1EGFRERBB2HDAC2HDAC6
SCHEMBL1065273 0.79 HDAC1 (0.71) HDAC1NAMPTEGFRHDAC3HDAC2
SCHEMBL1065274 0.79 HDAC1 (0.71) HDAC1NAMPTEGFRHDAC3HDAC2
SCHEMBL28469669 0.76 EGFR (0.61) HDAC1EGFRERBB2HDAC3HDAC2
SCHEMBL28146282 0.75 EGFR (0.68) HDAC1EGFRERBB2HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108409608-B Aromatic nitrogen mustard histone deacetylase inhibitor and preparation method and application thereof 潍坊医学院 2020-11-03 CN claimed
CN-108409608-B Aromatic nitrogen mustard histone deacetylase inhibitor and preparation method and application thereof 潍坊医学院 2020-11-03 CN disclosed