SCHEMBL28477323

SCHEMBL28477323

COc1cc(-n2c(=O)[nH]c3c(C(N)=O)nc(C4(OC)C=CC=CC4C(=O)O)cc32)cc(OC)c1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KATNA1 O75449 1/20 0.53
HSD17B10 Q99714 3/20 0.39
MAPT P10636 2/20 0.39
CSNK2A1 P68400 5/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
USP2 O75604 2/20 0.37
TSHR P16473 2/20 0.37
MAPK1 P28482 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 2/20 0.37
ESR1 P03372 1/20 0.37
TP53 P04637 1/20 0.37
HTT P42858 1/20 0.37
KDM4E B2RXH2 4/20 0.35
BRCA1 P38398 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30800070 0.72 KATNA1 (0.62) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL29176274 0.70 KATNA1 (0.80) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL30800011 0.70 KATNA1 (0.80) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL30800072 0.69 KATNA1 (1.00) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL29176296 0.69 KATNA1 (1.00) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL30799984 0.69 KATNA1 (0.82) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL29176303 0.69 KATNA1 (0.82) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL29176271 0.67 KATNA1 (0.73) KATNA1HSD17B10MAPTCSNK2A1CSNK2A2
SCHEMBL14149635 0.60 CSNK2A1 (0.68) HSD17B10MAPTCSNK2A1CSNK2A2CSNK2B
SCHEMBL29176297 0.56 MAP3K11 (0.44) KATNA1HSD17B10TP53KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111732584-A Diaryl substituted fused heterocyclic compound, preparation method thereof and application thereof in pharmacy 复旦大学 2020-10-02 CN disclosed