SCHEMBL28484352

SCHEMBL28484352

Cc1ccc2c(c(I)nn2C2CCCCO2)c1Br

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.38
CYP4A11 Q02928 3/20 0.38
GAA P10253 1/20 0.34
RET P07949 3/20 0.34
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
ATR Q13535 1/20 0.32
CYP2C19 P33261 1/20 0.32
ACVRL1 P37023 1/20 0.31
ACVR1 Q04771 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
ABL1 P00519 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
DGAT2 Q96PD7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30300121 1.00 CYP4F2 (0.38) CYP4F2CYP4A11GAARETRXRA
SCHEMBL24373243 0.88 GAA (0.41) CYP4F2CYP4A11GAARETRXRA
SCHEMBL29478900 0.88 GAA (0.41) CYP4F2CYP4A11GAARETRXRA
SCHEMBL30300226 0.85 CYP4F2 (0.38) CYP4F2CYP4A11GAARETRXRA
SCHEMBL21196075 0.85 CYP4F2 (0.38) CYP4F2CYP4A11GAARETRXRA
SCHEMBL24802947 0.82 CYP4F2 (0.36) CYP4F2CYP4A11GAARETRXRA
SCHEMBL20765166 0.81 CYP4F2 (0.35) CYP4F2CYP4A11RETRXRARXRB
SCHEMBL29936966 0.80 RET (0.35) CYP4F2CYP4A11GAARETRXRA
SCHEMBL26404733 0.80 RET (0.35) CYP4F2CYP4A11GAARETRXRA
SCHEMBL29937112 0.80 CYP4F2 (0.34) CYP4F2CYP4A11GAARETATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047937-B Tetrahydropyrido [3,4-d ] pyrimidin-2 (1H) -ones, their preparation and their pharmaceutical use 劲方医药科技(上海)有限公司 2023-04-07 CN disclosed
CN-112047937-A Tetrahydropyrido [3,4-d ] pyrimidin-2 (1H) -ones, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2020-12-08 CN disclosed