SCHEMBL28486407

SCHEMBL28486407

NC(=O)c1cccc2c1nc(-c1ccc(F)cc1)n2CCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.48
PKN1 Q16512 1/20 0.48
PKN2 Q16513 1/20 0.48
JAK2 O60674 2/20 0.43
JAK1 P23458 2/20 0.43
TYK2 P29597 2/20 0.43
JAK3 P52333 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PARP2 Q9UGN5 1/20 0.41
DHODH Q02127 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
TSSK1B Q9BXA7 2/20 0.39
MAPK14 Q16539 1/20 0.39
PIN1 Q13526 2/20 0.39
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29411959 1.00 PARP1 (0.48) PARP1PKN1PKN2JAK2JAK1
SCHEMBL28903059 0.90 HDAC1 (0.47) PARP1PKN1PKN2JAK2JAK1
SCHEMBL29411976 0.90 HDAC1 (0.47) PARP1PKN1PKN2JAK2JAK1
SCHEMBL28484147 0.87 PARP1 (0.51) PARP1PKN1PKN2MEN1KMT2A
SCHEMBL29411964 0.87 PARP1 (0.51) PARP1PKN1PKN2MEN1KMT2A
SCHEMBL28484710 0.85 HDAC1 (0.48) PARP1PKN1PKN2JAK2JAK1
SCHEMBL29411910 0.85 HDAC1 (0.48) PARP1PKN1PKN2JAK2JAK1
SCHEMBL28484826 0.84 PKN1 (0.48) PARP1PKN1PKN2JAK2JAK1
SCHEMBL29412003 0.84 PKN1 (0.48) PARP1PKN1PKN2JAK2JAK1
SCHEMBL29412030 0.82 CASR (0.47) PARP1PKN1PKN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111978301-A Benzimidazole compound with endothelial lipase inhibition effect and application thereof 盐城师范学院 2020-11-24 CN disclosed