SCHEMBL28487481

SCHEMBL28487481

O=C(NC1[CH]C1)c1cccc2ccn(Cc3ccc4ccccc4n3)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
FAAH O00519 3/20 0.40
TLR7 Q9NYK1 1/20 0.40
MCHR1 Q99705 2/20 0.39
HCRTR1 O43613 5/20 0.38
HCRTR2 O43614 4/20 0.38
PTGER4 P35408 2/20 0.37
PTGDR Q13258 2/20 0.37
TBXA2R P21731 1/20 0.37
PTGER1 P34995 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28494628 0.82 PTGER4 (0.37) HDAC1HDAC8HDAC6PTGER4PTGDR
SCHEMBL10085682 0.81 HDAC3 (0.44) HDAC11HDAC1HDAC3HDAC4HDAC7
SCHEMBL28486517 0.81 BCHE (0.43) HDAC11HDAC1HDAC3HDAC4HDAC7
SCHEMBL28487995 0.81 EGLN2 (0.39) HDAC11HDAC1HDAC3HDAC4HDAC7
SCHEMBL28487314 0.80 PTGER4 (0.35) HDAC1HDAC4HDAC6PTGER4PTGDR
SCHEMBL12583772 0.79 CYSLTR1 (0.47) HDAC11HDAC1HDAC3HDAC4HDAC7
SCHEMBL28493538 0.78 CBLB (0.34) PTGER4PTGDRTBXA2RPTGER1PTGFR
SCHEMBL28493532 0.78 PTGER4 (0.48) HDAC1HDAC3HDAC2HDAC10HDAC8
SCHEMBL28480177 0.78 KCNH2 (0.36) HDAC6PTGER4PTGDRTBXA2RPTGER1
SCHEMBL28484362 0.76 NPC1 (0.38) PTGER4PTGDRTBXA2RPTGER1PTGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111989311-B Compound for inhibiting PGE2/EP4 signal transduction, preparation method thereof and application thereof in medicines 凯复(苏州)生物医药有限公司 2022-03-22 CN disclosed
CN-111989311-A Compound for inhibiting PGE2/EP4 signal transduction, preparation method thereof and application thereof in medicines 凯复(苏州)生物医药有限公司 2020-11-24 CN disclosed