SCHEMBL28484362

SCHEMBL28484362

O=C(NC1[CH]C1)c1cccc2ccn(Cc3cc4ccccc4o3)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
MAOB P27338 2/20 0.38
PIN1 Q13526 1/20 0.38
RAB9A P51151 2/20 0.38
PTGER4 P35408 4/20 0.37
PTGDR Q13258 4/20 0.37
HTR1A P08908 1/20 0.37
HTR2B P41595 1/20 0.37
DRD2 P14416 2/20 0.37
DRD4 P21917 2/20 0.37
DRD3 P35462 2/20 0.37
CYP19A1 P11511 1/20 0.37
TBXA2R P21731 1/20 0.36
PTGER1 P34995 1/20 0.36
PTGFR P43088 1/20 0.36
PTGER3 P43115 1/20 0.36
PTGER2 P43116 1/20 0.36
STING1 Q86WV6 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28491847 0.89 HRH3 (0.38) PTGER4PTGDRHTR1AHTR2BTBXA2R
SCHEMBL28484335 0.89 CCR3 (0.36) PTGER4PTGDRTBXA2RPTGER1PTGFR
SCHEMBL28487960 0.88 CYP19A1 (0.39) NPC1MAOBPIN1RAB9AHTR1A
SCHEMBL28487995 0.82 EGLN2 (0.39) NPC1RAB9APTGER4PTGDRDRD2
SCHEMBL29518204 0.81 STING1 (0.48) NPC1MAOBRAB9APTGER4PTGDR
SCHEMBL12584456 0.81 STING1 (0.48) NPC1MAOBRAB9APTGER4PTGDR
SCHEMBL22276161 0.80 GPR52 (0.43) NPC1MAOBHTR1AHTR2BDRD2
SCHEMBL12584451 0.80 KDM4E (0.50) NPC1RAB9AHTR1AHTR2BDRD2
SCHEMBL30272259 0.79 PTGER4 (0.39) MAOBRAB9APTGER4PTGDRHTR1A
SCHEMBL987404 0.79 KDM4E (0.39) NPC1MAOBRAB9AHTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111989311-B Compound for inhibiting PGE2/EP4 signal transduction, preparation method thereof and application thereof in medicines 凯复(苏州)生物医药有限公司 2022-03-22 CN disclosed
CN-111989311-A Compound for inhibiting PGE2/EP4 signal transduction, preparation method thereof and application thereof in medicines 凯复(苏州)生物医药有限公司 2020-11-24 CN disclosed