SCHEMBL28488243

SCHEMBL28488243

CCOC(=O)C1=C(C)N(C)C(OCCCl)=C(C(=O)OC)C1c1ccccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.53
TSHR P16473 4/20 0.53
TP53 P04637 2/20 0.53
HTT P42858 2/20 0.53
TBXA2R P21731 3/20 0.52
ADRA1A P35348 3/20 0.52
SLC6A3 Q01959 3/20 0.52
HTR1A P08908 2/20 0.52
ADRA2A P08913 2/20 0.52
CHRM1 P11229 2/20 0.52
DRD1 P21728 2/20 0.52
SLC6A2 P23975 2/20 0.52
OPRM1 P35372 2/20 0.52
DRD3 P35462 2/20 0.52
KCNH2 Q12809 2/20 0.52
ABCB11 O95342 2/20 0.52
ABCB1 P08183 2/20 0.52
ADORA3 P0DMS8 2/20 0.52
ADRB3 P13945 2/20 0.52
OPRK1 P41145 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28497871 0.99 GAA (0.52) GAATSHRTP53HTTTBXA2R
SCHEMBL28403562 0.93 TBXA2R (0.58) GAATSHRTP53HTTTBXA2R
SCHEMBL6732477 0.93 TBXA2R (0.58) GAATSHRTP53HTTTBXA2R
SCHEMBL28488906 0.89 GAA (0.48) GAATSHRTP53HTTTBXA2R
SCHEMBL28356025 0.85 CYP2C9 (0.50) GAATSHRTP53HTTTBXA2R
SCHEMBL29259269 0.82 GAA (0.48) GAATSHRTP53HTTTBXA2R
SCHEMBL11130109 0.82 TBXA2R (0.42) GAATSHRTP53HTTTBXA2R
SCHEMBL14987090 0.81 TSHR (0.74) GAATSHRTP53HTTTBXA2R
SCHEMBL8199258 0.79 TSHR (0.73) GAATSHRTP53HTTTBXA2R
SCHEMBL19687545 0.79 TBXA2R (0.66) GAATSHRTP53HTTTBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010801-A Preparation method of amlodipine base 山东汇海医药化工有限公司 2020-12-01 CN claimed
CN-112010801-A Preparation method of amlodipine base 山东汇海医药化工有限公司 2020-12-01 CN disclosed