SCHEMBL28489176

SCHEMBL28489176

NC(Cc1cc(F)c(F)c(Cl)c1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.47
PTGS1 P23219 2/20 0.47
PKM P14618 2/20 0.47
ALPI P09923 1/20 0.47
XIAP P98170 1/20 0.47
GRIA2 P42262 1/20 0.47
USP2 O75604 3/20 0.45
ALOX15 P16050 3/20 0.45
HSD17B10 Q99714 3/20 0.45
TDP1 Q9NUW8 3/20 0.45
KDM4E B2RXH2 2/20 0.45
RECQL P46063 2/20 0.45
HIF1A Q16665 2/20 0.45
EGFR P00533 1/20 0.45
LCK P06239 1/20 0.45
FYN P06241 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
HTR2A P28223 1/20 0.45
PTGS2 P35354 1/20 0.45
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16095308 1.00 SLC7A5 (0.47) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL17596661 0.92 SLC7A5 (0.52) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL28485421 0.92 SLC7A5 (0.52) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL158046 0.88 SLC7A5 (0.55) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL158047 0.88 SLC7A5 (0.55) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL2130333 0.88 SLC7A5 (0.55) SLC7A5PTGS1PKMALPIXIAP
Hydrochloric Acid SCHEMBL1246362 0.86 SLC7A5 (0.53) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL15085642 0.86 GRIA2 (0.49) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL9951717 0.82 SLC7A5 (0.58) SLC7A5PTGS1PKMALPIXIAP
SCHEMBL9951720 0.82 SLC7A5 (0.58) SLC7A5PTGS1PKMALPIXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106999536-B Macrocyclic inhibitors of PD-1/PD-L1 and CD80(B7-1)/PD-L1 protein/protein interactions 百时美施贵宝公司 2020-11-27 CN disclosed