SCHEMBL28494337

SCHEMBL28494337

CN(C)/C=C/c1nc(C2CN(c3ccc([N+](=O)[O-])c(/C=C/N(C)C)n3)CCN2C(=O)OC(C)(C)C)ccc1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.39
NR1H2 P55055 6/20 0.36
NR1H3 Q13133 4/20 0.36
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
EIF2AK4 Q9P2K8 1/20 0.34
USP30 Q70CQ3 5/20 0.34
UCHL1 P09936 3/20 0.34
PRKCQ Q04759 1/20 0.34
HDAC1 Q13547 1/20 0.33
DPP4 P27487 1/20 0.33
TGM2 P21980 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12465844 0.83 MAPT (0.49) MAP4K4ALDH1A1MAPTLMNAPRKCQ
SCHEMBL12465843 0.83 MAPT (0.49) MAP4K4ALDH1A1MAPTLMNAPRKCQ
SCHEMBL30772278 0.83 MAPT (0.49) MAP4K4ALDH1A1MAPTLMNAPRKCQ
SCHEMBL30514215 0.83 USP30 (0.34) ALDH1A1MAPTLMNAUSP30UCHL1
SCHEMBL28488389 0.80 ALDH1A1 (0.37) MAP4K4ALDH1A1MAPTLMNA
SCHEMBL27930668 0.76 ALDH1A1 (0.37) ALDH1A1MAPTLMNA
SCHEMBL17461348 0.75 MAPT (0.40) ALDH1A1MAPT
SCHEMBL2338338 0.72 MAP4K4 (0.56) MAP4K4NR1H2NR1H3ALDH1A1MAPT
SCHEMBL2342450 0.72 MAP4K4 (0.56) MAP4K4NR1H2NR1H3ALDH1A1MAPT
SCHEMBL2338334 0.72 MAP4K4 (0.56) MAP4K4NR1H2NR1H3ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116942672-A Crystalline salts of B-RAF kinase inhibitors 徐诺药业公司 2023-10-27 CN disclosed
CN-111818924-B Crystalline salts of B-RAF kinase inhibitors 徐诺药业公司 2023-08-15 CN disclosed
CN-111818924-A Crystalline salts of B-RAF kinase inhibitors 徐诺药业公司 2020-10-23 CN disclosed