SCHEMBL28495014

SCHEMBL28495014

O=C(O)C1CCc2c(c3cc(OCc4ccccn4)ccc3n2C(=O)c2ccc(Cl)cc2)C1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.69
AKR1C2 P52895 3/20 0.69
PTGS1 P23219 3/20 0.69
AKR1C4 P17516 1/20 0.69
AKR1C1 Q04828 1/20 0.69
ALOX5 P09917 2/20 0.42
ALOX5AP P20292 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
EGFR P00533 1/20 0.42
IGF1R P08069 1/20 0.42
FLT4 P35916 1/20 0.42
KDR P35968 1/20 0.42
PARP10 Q53GL7 1/20 0.40
PTGS2 P35354 3/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
PPARG P37231 1/20 0.39
FFAR2 O15552 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28488499 0.89 AKR1C3 (0.74) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28500992 0.89 AKR1C3 (0.74) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28487851 0.89 AKR1C3 (0.74) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28496018 0.84 AKR1C3 (0.71) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL11836056 0.83 AKR1C3 (0.64) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL11834396 0.82 AKR1C3 (1.00) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28487853 0.82 AKR1C3 (0.68) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28074421 0.81 AKR1C3 (0.61) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28495383 0.80 PTGS1 (0.75) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL11844817 0.79 AKR1C3 (0.70) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN disclosed