SCHEMBL28500992

SCHEMBL28500992

O=C(O)[C@H]1CCc2c(c3cc(OCc4ccccc4)ccc3n2C(=O)c2ccc(Cl)cc2)C1

nearest known ligand 0.74

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.74
AKR1C2 P52895 3/20 0.74
PTGS1 P23219 3/20 0.74
AKR1C4 P17516 1/20 0.74
AKR1C1 Q04828 1/20 0.74
FFAR2 O15552 1/20 0.46
PTGS2 P35354 6/20 0.44
S1PR5 Q9H228 2/20 0.43
S1PR1 P21453 1/20 0.43
PRKX P51817 1/20 0.43
ACVR1 Q04771 1/20 0.43
PPARG P37231 2/20 0.42
PPARD Q03181 1/20 0.42
EGFR P00533 1/20 0.41
IGF1R P08069 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28487851 1.00 AKR1C3 (0.74) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28488499 1.00 AKR1C3 (0.74) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL11836056 0.94 AKR1C3 (0.64) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28074421 0.91 AKR1C3 (0.61) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28487853 0.90 AKR1C3 (0.68) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28495014 0.89 AKR1C3 (0.69) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL11837921 0.87 AKR1C3 (0.57) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28074596 0.86 AKR1C3 (0.54) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL28496018 0.86 AKR1C3 (0.71) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1
SCHEMBL11843978 0.86 AKR1C3 (0.54) AKR1C3AKR1C2PTGS1AKR1C4AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN claimed
CN-105646330-B Aromatic heterocyclic derivative and application thereof in medicine 贵州医科大学 2020-12-11 CN disclosed