SCHEMBL28495166

SCHEMBL28495166

Brc1ccc(-c2ccccc2-c2nccs2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.52
ABL1 P00519 1/20 0.47
BCR P11274 1/20 0.47
LOXL2 Q9Y4K0 1/20 0.42
CYP2A6 P11509 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
FBP1 P09467 1/20 0.40
RAB9A P51151 3/20 0.39
ADRB2 P07550 1/20 0.39
ADRA1A P35348 2/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1B P35368 1/20 0.39
NPC1 O15118 2/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
ADRA2A P08913 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
EDNRB P24530 1/20 0.38
EDNRA P25101 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2175845 0.85 PDPK1 (0.70) PDPK1LOXL2CYP2A6PTGDR2RAB9A
SCHEMBL5692672 0.83 PDPK1 (0.64) PDPK1LOXL2CYP2A6PTGDR2RAB9A
SCHEMBL8407091 0.83 PDPK1 (0.52) PDPK1LOXL2CYP2A6PTGDR2FBP1
SCHEMBL28487238 0.83 PDPK1 (0.52) PDPK1LOXL2CYP2A6PTGDR2FBP1
SCHEMBL9089977 0.83 PDPK1 (0.52) PDPK1LOXL2CYP2A6PTGDR2FBP1
SCHEMBL16990890 0.82 PDPK1 (0.56) PDPK1ABL1BCRLOXL2CYP2A6
SCHEMBL9086913 0.82 PDPK1 (0.51) PDPK1ABL1BCRLOXL2CYP2A6
SCHEMBL636877 0.81 PDPK1 (0.63) PDPK1ABL1BCRLOXL2CYP2A6
SCHEMBL1951149 0.81 PDPK1 (0.61) PDPK1LOXL2CYP2A6PTGDR2RAB9A
SCHEMBL28487118 0.80 ABL1 (0.42) PDPK1ABL1BCRLOXL2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111909110-A Preparation method of 2, 4-disubstituted thiazole compound 浙江工业大学 2020-11-10 CN disclosed