SCHEMBL28495237

SCHEMBL28495237

COc1ccc(CN2C(=O)C(F)(F)Oc3cc(F)c(N)cc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.43
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
SCN9A Q15858 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
CYP19A1 P11511 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
CHRM5 P08912 4/20 0.38
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
OPRL1 P41146 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30193840 0.87 CMA1 (0.43) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL25359325 0.87 CMA1 (0.43) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL26001081 0.84 SCN9A (0.39) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL28563929 0.83 CHRM5 (0.44) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL31478809 0.83 CMA1 (0.39) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL26001112 0.83 CHRM5 (0.39) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL25355571 0.82 SCN9A (0.38) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL25359029 0.81 CMA1 (0.38) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL25359718 0.80 PTPN1 (0.37) CMA1GSK3AGSK3BSCN9AL3MBTL1
SCHEMBL26001083 0.80 KDM4E (0.37) CMA1GSK3AGSK3BSCN9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727367-B Benzoxazinone compound containing pyridopyrimidinedione, preparation method and application thereof, and herbicide composition 山东先达农化股份有限公司 2021-01-05 CN disclosed
CN-110156767-B Cycloalkane pyrimidine diketone compound, preparation method and application thereof, and pesticide herbicide 南开大学 2020-12-11 CN disclosed