SCHEMBL28495366

SCHEMBL28495366

COc1cc(C(=O)O)c(N)c(OC)c1Br

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.54
FYN P06241 1/20 0.54
KDM4E B2RXH2 5/20 0.53
POLB P06746 1/20 0.53
PKM P14618 1/20 0.53
ALDH1A1 P00352 4/20 0.47
HSD17B10 Q99714 3/20 0.47
PTPN1 P18031 1/20 0.46
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
TSHR P16473 2/20 0.41
APOBEC3A P31941 1/20 0.41
HTT P42858 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GPR35 Q9HC97 1/20 0.40
GAA P10253 1/20 0.40
TPMT P51580 1/20 0.40
MYC P01106 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2034454 0.84 KDM4E (0.72) LCKFYNKDM4EPOLBPKM
SCHEMBL25165612 0.82 LCK (0.53) LCKFYNKDM4EPOLBPKM
SCHEMBL17494276 0.82 HSD17B10 (0.46) LCKFYNKDM4EPOLBPKM
SCHEMBL28270343 0.81 KDM4E (0.54) LCKFYNKDM4EPOLBPKM
SCHEMBL18669122 0.81 KDM4E (0.54) LCKFYNKDM4EPOLBPKM
SCHEMBL505418 0.81 LCK (0.56) LCKFYNKDM4EPKMALDH1A1
SCHEMBL31216003 0.79 LCK (0.53) LCKFYNKDM4EPOLBPKM
SCHEMBL28497490 0.78 PKM (0.76) LCKFYNKDM4EPOLBPKM
SCHEMBL642897 0.78 KDM4E (0.54) LCKFYNKDM4EPOLBPKM
SCHEMBL9197473 0.78 LCK (0.51) LCKFYNKDM4EPKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112110918-B Spiro substituted pyrimido cyclic compounds, process for their preparation and their use in medicine 劲方医药科技(上海)有限公司 2023-08-22 CN disclosed
CN-112110918-A Spiro-substituted pyrimido-cyclic compounds, preparation method and medical application thereof 劲方医药科技(上海)有限公司 2020-12-22 CN disclosed