SCHEMBL28496124

SCHEMBL28496124

O=C1O[C@@H](c2ccccc2)[C@@H](c2ccccc2)N(C(=O)O)[C@@H]1CCCC(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LIPG Q9Y5X9 3/20 0.33
NPC1 O15118 1/20 0.31
MDM2 Q00987 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30
MMP13 P45452 1/20 0.30
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18109442 0.86 ABCB1 (0.42) MDM2
SCHEMBL18109438 0.86 ABCB1 (0.42) MDM2
SCHEMBL19461020 0.86 ABCB1 (0.42) MDM2
SCHEMBL6063753 0.75 ELANE (0.36) MDM2
SCHEMBL6063582 0.75 ELANE (0.36) MDM2
SCHEMBL6918361 0.74 ELANE (0.35) PTGDR2
SCHEMBL22636048 0.74 ELANE (0.35) PTGDR2
SCHEMBL20134719 0.73 ABCB1 (0.43)
SCHEMBL18109300 0.73 ABCB1 (0.43)
SCHEMBL18109299 0.73 ABCB1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112174960-A Toll-like receptor modulating 4, 6-diamino-pyrido [3,2-D ] pyrimidine compounds 吉利德科学公司 2021-01-05 CN disclosed
CN-107108615-B Toll-like receptor modulating 4, 6-diamino-pyrido [3,2-D ] pyrimidine compounds 吉利德科学公司 2020-11-20 CN disclosed