SCHEMBL28500403

SCHEMBL28500403

Cc1nc(C(=O)NN)cn1C

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.47
MAPT P10636 3/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
KDM4E B2RXH2 6/20 0.40
ALDH1A1 P00352 7/20 0.39
GAA P10253 4/20 0.39
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.36
NPC1 O15118 1/20 0.36
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9710697 0.79 BRD4 (0.38) KDM4EALDH1A1POLBKMT2AL3MBTL1
SCHEMBL2551281 0.77 MAPT (0.49) P2RX7MAPTCYP1A2CYP3A4KDM4E
SCHEMBL8812476 0.76 SMN1; SMN2 (0.35) CYP1A2ALDH1A1POLBKMT2AL3MBTL1
SCHEMBL7489316 0.76 RXFP1 (0.42) MAPTKDM4EALDH1A1L3MBTL1
SCHEMBL15199632 0.76 MEN1 (0.41) CYP1A2CYP3A4KDM4EALDH1A1KMT2A
SCHEMBL16519359 0.73 CYP1A2 (0.53) MAPTCYP1A2KDM4EALDH1A1GAA
SCHEMBL21232986 0.71 MAPT (0.31) MAPT
SCHEMBL20713614 0.68
SCHEMBL22518496 0.68 P2RX7 (0.46) P2RX7MAPTCYP1A2CYP3A4KDM4E
SCHEMBL12911102 0.68 P2RX7 (0.42) P2RX7MAPTCYP1A2CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110105275-B Amide derivatives, preparation method and medical application thereof 上海海雁医药科技有限公司 2020-12-29 CN disclosed