SCHEMBL28501287

SCHEMBL28501287

COc1cc2nccc(Oc3ccc(Nc4c(NC5CC5)c(=O)c4=O)cc3)c2cc1C(N)=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 13/20 0.60
KDR P35968 5/20 0.58
AURKB Q96GD4 3/20 0.58
KIT P10721 3/20 0.58
PDGFRA P16234 3/20 0.58
FGFR2 P21802 3/20 0.58
PDGFRB P09619 2/20 0.58
FGFR1 P11362 2/20 0.58
FLT1 P17948 2/20 0.58
FLT4 P35916 2/20 0.58
AURKA O14965 2/20 0.58
MET P08581 2/20 0.58
TEK Q02763 2/20 0.58
RIPK2 O43353 1/20 0.58
ERN1 O75460 1/20 0.58
STK10 O94804 1/20 0.58
MAP3K6 O95382 1/20 0.58
ABL1 P00519 1/20 0.58
ESR1 P03372 1/20 0.58
ADORA3 P0DMS8 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29729414 0.88 RET (0.72) RETKDRAURKBKITPDGFRA
SCHEMBL28492935 0.88 RET (0.60) RETKDRAURKBKITPDGFRA
SCHEMBL19957132 0.88 RET (0.72) RETKDRAURKBKITPDGFRA
SCHEMBL28492198 0.86 RET (0.59) RETKDRAURKBKITPDGFRA
SCHEMBL19957010 0.85 RET (0.68) RETKDRAURKBKITPDGFRA
SCHEMBL28796987 0.84 FGFR2 (0.53) KDRAURKBKITPDGFRAFGFR2
SCHEMBL19956973 0.83 RET (0.65) RETKDRAURKBKITPDGFRA
SCHEMBL1249791 0.82 PDGFRA (0.77) RETKDRAURKBKITPDGFRA
SCHEMBL1892205 0.80 KDR (0.66) RETKDRAURKBKITPDGFRA
SCHEMBL12411989 0.78 KDR (0.65) RETKDRAURKBKITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892536-B Substituted quinoline carboxamides and their use 北京福元医药股份有限公司 2022-06-28 CN claimed
CN-111892536-A Substituted quinoline carboxamides and their use 北京福元医药股份有限公司 2020-11-06 CN claimed
CN-111892536-B Substituted quinoline carboxamides and their use 北京福元医药股份有限公司 2022-06-28 CN disclosed
CN-111892536-A Substituted quinoline carboxamides and their use 北京福元医药股份有限公司 2020-11-06 CN disclosed