SCHEMBL28501601

SCHEMBL28501601

CC(C)Oc1ccccc1-c1ccnc(N)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.59
CDK5R1 Q15078 5/20 0.59
CCNT1 O60563 3/20 0.59
CCNA2 P20248 3/20 0.59
CDK2 P24941 3/20 0.59
CDK9 P50750 3/20 0.59
CCNA1 P78396 3/20 0.59
CHRNA7 P36544 1/20 0.54
HSP90AA1 P07900 3/20 0.47
AURKA O14965 1/20 0.47
PRKACA P17612 1/20 0.47
ADORA2A P29274 1/20 0.47
GSK3B P49841 2/20 0.47
DYRK1A Q13627 2/20 0.47
HTR1A P08908 1/20 0.47
HTR7 P34969 1/20 0.47
HTR2B P41595 1/20 0.47
HTR5A P47898 1/20 0.47
NFATC1 O95644 1/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30507533 1.00 CDK5 (0.59) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL28506391 0.86 POLB (0.51) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL30507403 0.86 POLB (0.51) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL30507526 0.85 HSP90AA1 (0.47) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL28512809 0.85 HSP90AA1 (0.47) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL30507329 0.83 HSP90AA1 (0.60) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL3362587 0.83 HSP90AA1 (0.60) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL28506385 0.82 CHRNA7 (0.57) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL30507384 0.82 CHRNA7 (0.57) CDK5CDK5R1CCNT1CCNA2CDK2
SCHEMBL5470901 0.81 CCNT1 (0.55) CDK5CDK5R1CCNT1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-B Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2023-07-25 CN disclosed
CN-112010844-A Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2020-12-01 CN disclosed