SCHEMBL28502014

SCHEMBL28502014

Cc1cc(-c2cnc3[nH]cc(Br)c3c2)ccc1N1CCN(C)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 6/20 0.58
IL2 P60568 3/20 0.47
MAP3K11 Q16584 7/20 0.45
DYRK1A Q13627 1/20 0.44
TNIK Q9UKE5 8/20 0.44
IKBKB O14920 2/20 0.41
CHUK O15111 2/20 0.41
ABL1 P00519 2/20 0.41
INSR P06213 2/20 0.41
CDK2 P24941 2/20 0.41
FLT3 P36888 2/20 0.41
SGK1 O00141 1/20 0.40
AURKA O14965 1/20 0.40
PRKAB2 O43741 1/20 0.40
ROCK2 O75116 1/20 0.40
NTRK1 P04629 1/20 0.40
LCK P06239 1/20 0.40
CDK1 P06493 1/20 0.40
IGF1R P08069 1/20 0.40
MET P08581 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499901 0.87 MAP4K1 (0.61) MAP4K1IL2MAP3K11DYRK1ATNIK
SCHEMBL28506939 0.86 MAP4K1 (0.47) MAP4K1IL2MAP3K11DYRK1ATNIK
SCHEMBL31536249 0.86 MAP4K1 (0.47) MAP4K1IL2MAP3K11DYRK1ATNIK
SCHEMBL28513907 0.86 ROCK2 (0.48) MAP4K1IL2DYRK1ATNIKROCK2
SCHEMBL28504488 0.86 MAP4K1 (0.59) MAP4K1IL2MAP3K11DYRK1A
SCHEMBL28499623 0.84 CHEK1 (0.46) MAP4K1IL2MAP3K11DYRK1ATNIK
SCHEMBL21590290 0.84 MAP4K1 (0.64) MAP4K1IL2TNIK
SCHEMBL28504384 0.82 MAP4K1 (0.66) MAP4K1IL2MAP3K11TNIKIKBKB
SCHEMBL28506141 0.82 MAP4K1 (0.46) MAP4K1IL2MAP3K11DYRK1AABL1
SCHEMBL21592600 0.81 MAP3K11 (0.66) MAP4K1IL2MAP3K11DYRK1ATNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed