SCHEMBL28503231

SCHEMBL28503231

Cc1cc(-c2cnc3[nH]ccc3c2)ccc1C1=CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 4/20 0.56
PIK3CA P42336 1/20 0.47
BRD4 O60885 1/20 0.45
CDK9 P50750 3/20 0.45
WNT3A P56704 1/20 0.45
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB1 P18505 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44
GABRA4 P48169 1/20 0.44
GABRE P78334 1/20 0.44
GABRA6 Q16445 1/20 0.44
GABRG1 Q8N1C3 1/20 0.44
GABRG3 Q99928 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15560997 0.91 JAK1 (0.55) JAK1PIK3CABRD4CDK9WNT3A
SCHEMBL28499853 0.87 PLK4 (0.45) JAK1PIK3CACDK9CCNT1CDK7
SCHEMBL21590284 0.80 JAK1 (0.43) JAK1BRD4CDK9WNT3AGABRP
SCHEMBL28507487 0.80 MAP4K1 (0.51) JAK1CDK9GABRPGABRDGABRA1
SCHEMBL20112166 0.79 PDK4 (0.58) JAK1GABRPGABRDGABRA1GABRB1
SCHEMBL15778686 0.78 ESR2 (0.54) JAK1PIK3CABTKCDK7CDK8
SCHEMBL15778894 0.78 NR1H2 (0.53) JAK1PIK3CABTKCDK7CDK8
SCHEMBL28906243 0.78 HTR6 (0.42) JAK1CDK9WNT3AGABRPGABRD
SCHEMBL27025890 0.78 GRM1 (0.51) JAK1GABRPGABRDGABRA1GABRB1
SCHEMBL31198348 0.76 BCL2 (0.58) JAK1BRD4CDK9CYP11B2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed