SCHEMBL28504378

SCHEMBL28504378

Cc1cc(-c2cnc3[nH]cc(-c4ccnc(C(=O)O)n4)c3c2)ccc1N1CCN(C)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 5/20 0.56
DYRK1A Q13627 1/20 0.47
CAMKK2 Q96RR4 1/20 0.46
KMO O15229 2/20 0.46
CCNT1 O60563 6/20 0.44
CCNA2 P20248 6/20 0.44
CDK2 P24941 6/20 0.44
CDK9 P50750 6/20 0.44
MAP3K11 Q16584 3/20 0.44
IL2 P60568 3/20 0.44
TNIK Q9UKE5 1/20 0.43
PIK3CG P48736 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21593047 0.91 MAP4K1 (0.54) MAP4K1DYRK1ACCNT1CCNA2CDK2
SCHEMBL28502252 0.84 MAP4K1 (0.65) MAP4K1CAMKK2MAP3K11IL2TNIK
SCHEMBL28511323 0.81 MAP4K1 (0.55) MAP4K1DYRK1ACAMKK2CDK2MAP3K11
Hydrochloric Acid SCHEMBL28507116 0.80 MAP4K1 (0.54) MAP4K1DYRK1ACAMKK2MAP3K11IL2
SCHEMBL28511448 0.79 MAP4K1 (0.63) MAP4K1CAMKK2MAP3K11IL2TNIK
SCHEMBL21592665 0.79 MAP4K1 (0.55) MAP4K1DYRK1ACAMKK2MAP3K11IL2
SCHEMBL21592647 0.78 MAP4K1 (0.62) MAP4K1CAMKK2MAP3K11IL2TNIK
SCHEMBL21592622 0.78 MAP4K1 (0.59) MAP4K1CAMKK2MAP3K11IL2TNIK
SCHEMBL28504384 0.77 MAP4K1 (0.66) MAP4K1CDK2MAP3K11IL2TNIK
SCHEMBL21593022 0.77 MAP4K1 (0.61) MAP4K1DYRK1ACAMKK2MAP3K11IL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed