SCHEMBL28508013

SCHEMBL28508013

NC(=O)OCCC(O)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.49
AOC3 Q16853 1/20 0.44
GAA P10253 1/20 0.41
GABBR2 O75899 5/20 0.39
GABBR1 Q9UBS5 5/20 0.39
LMNA P02545 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2D6 P10635 3/20 0.39
CYP2C19 P33261 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP3A4 P08684 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
NFKB1 P19838 1/20 0.39
DRD3 P35462 1/20 0.39
BLM P54132 1/20 0.39
THRB P10828 1/20 0.39
TSHR P16473 1/20 0.39
CHRNB2 P17787 2/20 0.39
CHRNB4 P30926 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28508012 1.00 CYP1A2 (0.49) CYP1A2AOC3GAAGABBR2GABBR1
SCHEMBL28513886 1.00 CYP1A2 (0.49) CYP1A2AOC3GAAGABBR2GABBR1
SCHEMBL18548754 0.83 SMN1; SMN2 (0.56) CYP1A2AOC3LMNACYP2D6CHRNB2
SCHEMBL25216149 0.81 ADRB3 (0.43) CYP1A2CYP2D6MEN1KMT2AL3MBTL1
SCHEMBL28507778 0.80 AOC3 (0.49) CYP1A2AOC3CHRNB2CHRNB4CHRNA3
SCHEMBL28505084 0.80 AOC3 (0.49) CYP1A2AOC3CHRNB2CHRNB4CHRNA3
SCHEMBL28505083 0.80 AOC3 (0.49) CYP1A2AOC3CHRNB2CHRNB4CHRNA3
SCHEMBL21462735 0.78 TDP1 (0.53) CYP1A2GAALMNACYP2D6CYP2C19
SCHEMBL21462737 0.78 TDP1 (0.53) CYP1A2GAALMNACYP2D6CYP2C19
SCHEMBL27953236 0.76 MAPT (0.43) AOC3GAAMEN1KMT2ACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112262139-B Aminopyrrolotriazines as kinase inhibitors 百时美施贵宝公司 2023-07-25 CN disclosed
CN-112262139-A Aminopyrrolotriazines as kinase inhibitors 百时美施贵宝公司 2021-01-22 CN disclosed