SCHEMBL28505083

SCHEMBL28505083

CO[C@@H](CCOC(N)=O)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.49
CYP1A2 P05177 1/20 0.46
UTS2R Q9UKP6 7/20 0.40
CHRNB2 P17787 2/20 0.39
CHRNB4 P30926 2/20 0.39
CHRNA3 P32297 2/20 0.39
CHRNA4 P43681 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28507778 1.00 AOC3 (0.49) AOC3CYP1A2UTS2RCHRNB2CHRNB4
SCHEMBL28505084 1.00 AOC3 (0.49) AOC3CYP1A2UTS2RCHRNB2CHRNB4
SCHEMBL28508012 0.80 CYP1A2 (0.49) AOC3CYP1A2CHRNB2CHRNB4CHRNA3
SCHEMBL28513886 0.80 CYP1A2 (0.49) AOC3CYP1A2CHRNB2CHRNB4CHRNA3
SCHEMBL28508013 0.80 CYP1A2 (0.49) AOC3CYP1A2CHRNB2CHRNB4CHRNA3
SCHEMBL3685753 0.79 AOC3 (0.54) AOC3UTS2R
SCHEMBL3685751 0.79 AOC3 (0.54) AOC3UTS2R
SCHEMBL639174 0.76 AOC3 (0.49) AOC3CYP1A2UTS2R
SCHEMBL21199033 0.75 AOC3 (0.59) AOC3UTS2RCHRNB2CHRNA4
SCHEMBL21198899 0.75 AOC3 (0.59) AOC3UTS2RCHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112262139-B Aminopyrrolotriazines as kinase inhibitors 百时美施贵宝公司 2023-07-25 CN disclosed
CN-112262139-A Aminopyrrolotriazines as kinase inhibitors 百时美施贵宝公司 2021-01-22 CN disclosed