SCHEMBL28508016

SCHEMBL28508016

Cc1[c]cccc1-n1ccnn1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 15/20 0.44
KEAP1 Q14145 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CHRNB2 P17787 1/20 0.36
CYP2B6 P20813 1/20 0.36
MAOA P21397 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRNA4 P43681 1/20 0.36
HTR3A P46098 1/20 0.36
EGLN2 Q96KS0 1/20 0.35
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28506122 0.77 MAPK1 (0.46) NOTUMHCRTR1HCRTR2
SCHEMBL28511732 0.76 ALDH1A1 (0.47) NOTUM
SCHEMBL1586846 0.76 NOTUM (0.44) NOTUMKEAP1EGLN2HCRTR1HCRTR2
SCHEMBL241942 0.74 NOTUM (0.50) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL16113420 0.71 NOTUM (0.47) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL18378736 0.71 NOTUM (0.47) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL28509696 0.71
SCHEMBL9685417 0.70 GAA (0.40) CYP1A2CYP2C19
SCHEMBL586173 0.69 NOTUM (0.40) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL1836207 0.69 IDO1 (0.50) NOTUMCYP1A2CYP2C9CYP2C19CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026067-B 6-amino-quinoline-3-carbonitriles as COT modulators 吉利德科学公司 2021-01-12 CN disclosed