SCHEMBL28508665

SCHEMBL28508665

CC1(O)CCN(C(=O)c2ccc(B(O)O)cc2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM3 Q14832 1/20 0.47
GPR183 P32249 1/20 0.45
HSD17B10 Q99714 4/20 0.40
CYP2C9 P11712 3/20 0.40
CYP2D6 P10635 3/20 0.40
USP2 O75604 1/20 0.40
TSHR P16473 1/20 0.40
VNN1 O95497 1/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C19 P33261 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40
GABRA2 P47869 1/20 0.40
GABRB2 P47870 1/20 0.40
GABRA4 P48169 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25668251 0.81 CRBN (0.54) GRM3CYP2C9CYP2D6TSHRCYP2C19
SCHEMBL951459 0.81 NAMPT (0.53) GPR183HSD17B10CYP2C9CYP3A4CYP2C19
SCHEMBL29950978 0.77 HPGD (0.57) ALDH1A1HPGDPKMPOLB
SCHEMBL31037268 0.77 GPR183 (0.47) GPR183TSHRGABRDGABRA1GABRB1
SCHEMBL204078 0.74 HPGD (0.70) USP2TSHRALDH1A1HPGD
SCHEMBL950365 0.74 HPGD (0.64) HSD17B10TSHRALDH1A1HPGDPOLB
SCHEMBL15758020 0.73 GPR183 (0.44) GPR183TSHRALDH1A1HPGDPKM
SCHEMBL532147 0.73 POLB (0.65) CYP2C9CYP2D6TSHRCYP2C19HPGD
SCHEMBL15473398 0.73 GABRD (0.63) GRM3GABRDGABRA1GABRB1GABRA5
SCHEMBL28502409 0.73 GPR183 (0.46) GPR183HSD17B10CYP2C9CYP2D6USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed