SCHEMBL28508666

SCHEMBL28508666

Cc1cc(-c2cnc3[nH]cc(-c4ccc(C(N)=O)c(C)c4C)c3c2)ccc1C1CCN(C)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 10/20 0.49
MAP4K1 Q92918 3/20 0.48
IL2 P60568 1/20 0.48
MAP3K11 Q16584 4/20 0.47
AURKA O14965 2/20 0.45
SGK2 Q9HBY8 2/20 0.45
SGK1 O00141 1/20 0.45
CAMKK1 Q8N5S9 1/20 0.45
SGK3 Q96BR1 1/20 0.45
PIK3CG P48736 2/20 0.45
CDC7 O00311 1/20 0.43
PLK4 O00444 1/20 0.43
CHEK1 O14757 1/20 0.43
MAPK13 O15264 1/20 0.43
PDPK1 O15530 1/20 0.43
DYRK3 O43781 1/20 0.43
ROCK2 O75116 1/20 0.43
RPS6KA5 O75582 1/20 0.43
PRKD3 O94806 1/20 0.43
PAK4 O96013 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28501998 0.90 CAMKK2 (0.48) CAMKK2MAP4K1IL2MAP3K11AURKA
SCHEMBL28514859 0.90 CAMKK2 (0.50) CAMKK2MAP3K11AURKASGK2SGK1
SCHEMBL28906202 0.90 CAMKK2 (0.54) CAMKK2MAP4K1IL2MAP3K11AURKA
SCHEMBL28510111 0.86 MAP4K1 (0.55) CAMKK2MAP4K1IL2MAP3K11AURKA
SCHEMBL28506325 0.85 MAP4K1 (0.57) CAMKK2MAP4K1IL2MAP3K11AURKA
SCHEMBL28502218 0.83 MAP4K1 (0.54) CAMKK2MAP4K1IL2MAP3K11PIK3CG
SCHEMBL28597669 0.82 PAK1 (0.58) CAMKK2MAP4K1IL2MAP3K11AURKA
SCHEMBL28513743 0.82 MAP4K1 (0.60) CAMKK2MAP4K1IL2MAP3K11CHEK1
SCHEMBL28605051 0.81 PAK1 (0.58) CAMKK2MAP4K1IL2MAP3K11AURKA
SCHEMBL28499626 0.81 MAP4K1 (0.61) CAMKK2MAP4K1IL2MAP3K11CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed