SCHEMBL28512125

SCHEMBL28512125

CCCCS(=O)(=O)Nc1ccc(B2OC(C)(C)C(C)(C)O2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.61
CA2 P00918 5/20 0.61
CA9 Q16790 5/20 0.61
CA12 O43570 1/20 0.61
CA3 P07451 1/20 0.61
CA4 P22748 1/20 0.61
CA6 P23280 1/20 0.61
CA5A P35218 1/20 0.61
CA7 P43166 1/20 0.61
CA14 Q9ULX7 1/20 0.61
CA5B Q9Y2D0 1/20 0.61
LPL P06858 6/20 0.51
LIPG Q9Y5X9 6/20 0.51
HPGD P15428 2/20 0.49
LMNA P02545 1/20 0.49
BRD4 O60885 1/20 0.47
AR P10275 1/20 0.46
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12707453 0.92 CA1 (0.64) CA1CA2CA9CA12CA3
SCHEMBL24133598 0.87 CA1 (0.69) CA1CA2CA9CA12CA3
SCHEMBL488760 0.83 CA1 (0.57) CA1CA2CA9CA12CA3
SCHEMBL488838 0.82 CA1 (0.59) CA1CA2CA9CA12CA3
SCHEMBL23281878 0.80 CA1 (0.57) CA1CA2CA9CA12CA3
SCHEMBL15091838 0.80 CA1 (0.43) CA1CA2CA9CA12CA3
SCHEMBL15649561 0.79 BRD4 (0.39) CA1CA2CA9CA12CA3
SCHEMBL488832 0.78 CA1 (0.54) CA1CA2CA9CA12CA3
SCHEMBL488897 0.78 CA1 (0.54) CA1CA2CA9CA12CA3
SCHEMBL1560571 0.78 CA1 (0.61) CA1CA2CA9CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed