SCHEMBL28512236

SCHEMBL28512236

Cn1cc(-c2cnc3[nH]cc(Br)c3c2)cn1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 15/20 0.54
PDPK1 O15530 4/20 0.53
TNIK Q9UKE5 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL720228 0.83 ALK (0.57) ALKPDPK1TNIK
SCHEMBL16344211 0.83 PDPK1 (0.58) ALKPDPK1
SCHEMBL28506207 0.82 ALK (0.48) ALKPDPK1
SCHEMBL28503574 0.81 PAK1 (0.56) PDPK1TNIK
SCHEMBL9888143 0.80 ALK (0.51) ALKPDPK1TNIK
SCHEMBL9284633 0.80 ALK (0.56) ALKPDPK1
SCHEMBL9278508 0.80 ALK (0.54) ALKPDPK1TNIK
SCHEMBL15253627 0.79 ALK (0.48) ALKPDPK1
SCHEMBL28481416 0.78 PDPK1 (0.51) ALKPDPK1
SCHEMBL9887923 0.77 ALK (0.48) ALKPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed