SCHEMBL28503574

SCHEMBL28503574

CN1CCC(n2cc(-c3cnc4[nH]cc(Br)c4c3)cn2)CC1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 12/20 0.56
TNIK Q9UKE5 1/20 0.53
MET P08581 4/20 0.50
PAK4 O96013 3/20 0.50
IKBKE Q14164 1/20 0.48
TBK1 Q9UHD2 1/20 0.48
SIK1 P57059 1/20 0.48
SIK3 Q9Y2K2 1/20 0.48
PDPK1 O15530 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28512236 0.81 ALK (0.54) TNIKPDPK1
SCHEMBL21592674 0.80 MAP3K11 (0.61) PAK1TNIKPAK4SIK1SIK3
SCHEMBL31435909 0.79 TNIK (0.55) PAK1TNIKPAK4SIK1SIK3
SCHEMBL19860027 0.78 SIK1 (0.65) PAK1TNIKMETPAK4SIK1
SCHEMBL21776509 0.78 MET (0.55) METIKBKETBK1
SCHEMBL30388408 0.78 MET (0.55) METIKBKETBK1
SCHEMBL28502521 0.77 DYRK1A (0.64) PAK1TNIKMETIKBKETBK1
SCHEMBL15799467 0.76 SIK1 (0.82) PAK1TNIKMETPAK4SIK1
SCHEMBL15799697 0.76 TNIK (0.52) PAK1TNIKMETPAK4SIK1
SCHEMBL21626734 0.76 MET (0.56) PAK1TNIKMETPAK4SIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed